Synthesis of Amides Based on Biologically Active 5Z,9Z-Eicosadienoic Acid

Мұқаба

Дәйексөз келтіру

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Аннотация

For the first time, amides of (5Z,9Z)-eicosa-5,9-dienoic acid, which exhibits a high inhibitory activity of topoisomerases I and II, were synthesized using aliphatic and O-containing 1,2-dienes at the key stage of the intermolecular cross-cyclomagnesiation reaction, catalyzed by Cp2TiCl2.

Толық мәтін

Рұқсат жабық

Авторлар туралы

E. Makarova

Institute of Petrochemistry and Catalysis of the Ufa Federal Research Center of the Russian Academy of Sciences

Хат алмасуға жауапты Автор.
Email: makarovaelina87@gmail.com
ORCID iD: 0000-0001-7481-0880
Ресей, 141, Oktyabr Ave., Ufa, 450075

A. Makarov

Institute of Petrochemistry and Catalysis of the Ufa Federal Research Center of the Russian Academy of Sciences

Email: makarovaelina87@gmail.com
ORCID iD: 0000-0001-7870-2334
Ресей, 141, Oktyabr Ave., Ufa, 450075

U. Dzhemilev

Zelinsky Institute of Organic Chemistry of the Russian Academy of Sciences

Email: makarovaelina87@gmail.com
ORCID iD: 0000-0002-7992-6337
Ресей, 47, Leninsky Ave., Moscow, 119991

V. Dyakonov

Zelinsky Institute of Organic Chemistry of the Russian Academy of Sciences

Email: makarovaelina87@gmail.com
ORCID iD: 0000-0002-7787-5054
Ресей, 47, Leninsky Ave., Moscow, 119991

Әдебиет тізімі

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3. Scheme 1

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